Discovery of structurally distinct tricyclic M positive allosteric modulator (PAM) chemotypes
AUTHORS
Temple
KJKayla J ,
Long
MFMadeline F ,
Engers
JLJulie L ,
Watson
KJKatherine J ,
Chang
SSichen ,
Luscombe
VBVincent B ,
Rodriguez
ALAlice L ,
Niswender
CMColleen M ,
Bridges
TMThomas M ,
Conn
PJP Jeffrey ,
Engers
DWDarren W ,
Lindsley
CWCraig W .
Bioorganic & medicinal chemistry letters. 2019 11 11; 30(4).
126811
- PMID: 31787491[PubMed].
ABSTRACT
Tags: 2019